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Home > Category > > Small Molecule Compound > CH6953755

CH6953755

Glpbio
Catalog No:GC39557-10mM (in 1mL DMSO) CAS No.:2055918-71-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:CH6953755 是一種有效的,具有口服活性和選擇性的 YES1 激酶 (SRC 家族的成員)抑制劑,IC50 為 1.8 nM。CH6953755 通過(guò)抑制 YES1 激酶,從而在體內(nèi)外對(duì) YES1 基因擴(kuò)增的癌癥產(chǎn)生抗腫瘤活性。DMSO: 125 mg/mL (226.22 mM)
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